Abstract
Dihydro-oxadiazine and its derivatives have been demonstrated to be important heterocyclic scaffold platform with bioactive diversity, which present wide activities such as cardiovascular, antitumor, antibacterial, antimicrobial, acricidal, insecticidal, plant-growth regulating, chitin biosynthesis inhibitors and monoamine oxidase inhibition. Versatile features of dihydro-oxadiazine heterocycles have emerged, so the aim of the present paper was to review the recent advances of dihydro-oxadiazine-based heterocyclic derivatives mainly including synthesis and biological activities.
Keywords: Dihydro-oxadiazine, heterocycle, synthesis, biological activity, heterocyclic scaffold, cardiovascular, antitumor, antibacterial, antimicrobial, acricidal, insecticidal, plant-growth regulating, chitin biosynthesis, monoamine oxidase
Mini-Reviews in Medicinal Chemistry
Title: Synthesis and Biological Properties of Dihydro-Oxadiazine-Based Heterocyclic Derivatives
Volume: 11 Issue: 8
Author(s): S. Ke, X. Cao, Y. Liang, K. Wang and Z. Yang
Affiliation:
Keywords: Dihydro-oxadiazine, heterocycle, synthesis, biological activity, heterocyclic scaffold, cardiovascular, antitumor, antibacterial, antimicrobial, acricidal, insecticidal, plant-growth regulating, chitin biosynthesis, monoamine oxidase
Abstract: Dihydro-oxadiazine and its derivatives have been demonstrated to be important heterocyclic scaffold platform with bioactive diversity, which present wide activities such as cardiovascular, antitumor, antibacterial, antimicrobial, acricidal, insecticidal, plant-growth regulating, chitin biosynthesis inhibitors and monoamine oxidase inhibition. Versatile features of dihydro-oxadiazine heterocycles have emerged, so the aim of the present paper was to review the recent advances of dihydro-oxadiazine-based heterocyclic derivatives mainly including synthesis and biological activities.
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Cite this article as:
Ke S., Cao X., Liang Y., Wang K. and Yang Z., Synthesis and Biological Properties of Dihydro-Oxadiazine-Based Heterocyclic Derivatives, Mini-Reviews in Medicinal Chemistry 2011; 11 (8) . https://dx.doi.org/10.2174/138955711796268769
DOI https://dx.doi.org/10.2174/138955711796268769 |
Print ISSN 1389-5575 |
Publisher Name Bentham Science Publisher |
Online ISSN 1875-5607 |
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