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Preparative Synthesis of 7-Carboxy-2-R-isoindol-1-ones

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

A preparative method for the synthesis of 7-carboxy-2-R-isoindol-1-ones was developed on the basis of the [4+2] cycloaddition of secondary furfurylamines to maleic anhydride.

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Varlamov, A.V., Boltukhina, E.V., Zubkov, F.I. et al. Preparative Synthesis of 7-Carboxy-2-R-isoindol-1-ones. Chemistry of Heterocyclic Compounds 40, 22–28 (2004). https://doi.org/10.1023/B:COHC.0000023763.75894.63

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  • DOI: https://doi.org/10.1023/B:COHC.0000023763.75894.63

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